Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50022606
Affinity DataKi: 4.60nMAssay Description:Competitive inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex assessed as inhibition constant in presence of cofactor SA...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of wild type EZH2 methyltransferase activity (unknown origin) using 3H-SAM as substrate incubated for 30 mins by Microscint-O scintillatio...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of EZH2 Y641F mutant (unknown origin) using HMT as substrate incubated for 60 mins by luminescence based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of EZH1 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human EZH2 using histone H1 as substrate incubated for 30 mins followed by substrate addition and measured after 90 mins by Microscint-...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of human EZH2 in human MCF-10A cells assessed as reduction in H3K27me3 levels incubated for 72 hrs by In-cell western assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity to H3 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity to NET (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of EZH2 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of EZH1 methyltransferase activity (unknown origin) in PRC2 complex using 3H-SAM as substrate by Scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of G9a (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SMYD2 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SETD7 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SETD8 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SUV39H2 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SUV420H1 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT1 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MLL1 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT3 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of DOT1L (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EHMT1 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SUV420H2 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of DNMT1 (unknown origin) using hemimethylated dsDNA as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SETDB1 (unknown origin) using [3H-SAM] as substrate incubated for 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of EZH2 Y641F mutant (unknown origin) using HMT as substrate incubated for 60 mins by luminescence based analysisMore data for this Ligand-Target Pair
