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Found 20 Enz. Inhib. hit(s) with all data for entry = 50042981
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434151(CHEMBL2381666)
Affinity DataKi:  22nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434153(CHEMBL2381668)
Affinity DataKi:  24nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434152(CHEMBL2381665)
Affinity DataKi:  43nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434148(CHEMBL2381663)
Affinity DataKi:  52nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434147(CHEMBL2381661)
Affinity DataKi:  61nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434145(CHEMBL2381660)
Affinity DataKi:  64nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMpH: 7.8Assay Description:Inhibition of PSA (unknown origin) in 50 mM TRIS.HCL and 100 mM NaCl buffer at pH 7.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434146(CHEMBL2381670)
Affinity DataKi:  73nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  75nMAssay Description:Inhibition of PSA (unknown origin) in RPMIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434143(CHEMBL2381658)
Affinity DataKi:  102nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  142nMAssay Description:Inhibition of PSA (unknown origin) in RPMI in presence of 1% fetal bovine serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434154(CHEMBL2381667)
Affinity DataKi:  165nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434144(CHEMBL2381659)
Affinity DataKi:  229nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434150(CHEMBL2381664)
Affinity DataKi:  302nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434149(CHEMBL2381662)
Affinity DataKi:  310nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  604nMAssay Description:Inhibition of PSA (unknown origin) in female plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  699nMAssay Description:Inhibition of PSA (unknown origin) in RPMI in presence of 1% fetal bovine serum, 1% penicillin/streptomycin, 1% L-glutamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434141(CHEMBL2381657)
Affinity DataKi:  4.50E+4nMAssay Description:Inhibition of PSA (unknown origin) using Mu-SRKSQQY-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50099216((2S,3S)-1-[2-(3-Benzyloxycarbonyl-phenyl)-acetyl]-...)
Affinity DataIC50:  226nMAssay Description:Inhibition of PSA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed