Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50043117
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436224BDBM50436224(CHEMBL2398697)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436223BDBM50436223(CHEMBL2398698)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436222BDBM50436222(CHEMBL2398699)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436244BDBM50436244(CHEMBL2398669)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436236BDBM50436236(CHEMBL2398678)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human SK-Mel-147 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436221BDBM50436221(CHEMBL2398700)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436255BDBM50436255(CHEMBL2398701)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436236BDBM50436236(CHEMBL2398678)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436241BDBM50436241(CHEMBL2398672)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436254BDBM50436254(CHEMBL2398702)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436243BDBM50436243(CHEMBL2398670)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436237BDBM50436237(CHEMBL603141)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436235BDBM50436235(CHEMBL2398679)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436239BDBM50436239(CHEMBL2398674)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436240BDBM50436240(CHEMBL2398673)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436253BDBM50436253(CHEMBL2398703)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436252BDBM50436252(CHEMBL2398704)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436251BDBM50436251(CHEMBL2398705)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436242BDBM50436242(CHEMBL2398671)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436250BDBM50436250(CHEMBL2398706)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436233BDBM50436233(CHEMBL2398681)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436234BDBM50436234(CHEMBL2398680)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436249BDBM50436249(CHEMBL2398707)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436238BDBM50436238(CHEMBL2398676)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436247BDBM50436247(CHEMBL2398709)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436248BDBM50436248(CHEMBL2398708)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436232BDBM50436232(CHEMBL2398682)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436231BDBM50436231(CHEMBL2398683)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436230BDBM50436230(CHEMBL2398684)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436229BDBM50436229(CHEMBL2398685)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436228BDBM50436228(CHEMBL2398686)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436227BDBM50436227(CHEMBL2398687)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436246BDBM50436246(CHEMBL2398710)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436226BDBM50436226(CHEMBL2398688)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436245BDBM50436245(CHEMBL2398711)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTransforming protein RhoA(Human)
College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50436225BDBM50436225(CHEMBL2398689)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of RhoC-mediated pathway in human PC3 cells assessed as inhibition of SRE-regulated gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed