Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50043155
TargetAurora kinase A(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM52755(MLS001004059 | N-[2-(2-cyano-4-nitro-anilino)ethyl...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of Aurora A kinase (unknown origin) by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM52755(MLS001004059 | N-[2-(2-cyano-4-nitro-anilino)ethyl...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of Aurora B kinase (unknown origin) by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM52755(MLS001004059 | N-[2-(2-cyano-4-nitro-anilino)ethyl...)
Affinity DataIC50:  141nMAssay Description:Inhibition of recombinant Aurora B kinase (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed