Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50043277
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438573BDBM50438573(CHEMBL2413705)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438573BDBM50438573(CHEMBL2413705)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438581BDBM50438581(CHEMBL448807)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438581BDBM50438581(CHEMBL448807)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438576BDBM50438576(CHEMBL2413704)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438567BDBM50438567(CHEMBL512713)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438568BDBM50438568(CHEMBL2413710)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438575BDBM50438575(CHEMBL486977)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438576BDBM50438576(CHEMBL2413704)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438566BDBM50438566(CHEMBL2413711)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438568BDBM50438568(CHEMBL2413710)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438574BDBM50438574(CHEMBL486969)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438571BDBM50438571(CHEMBL2413707)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438580BDBM50438580(CHEMBL2413700)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438575BDBM50438575(CHEMBL486977)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438580BDBM50438580(CHEMBL2413700)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438579BDBM50438579(CHEMBL2413701)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438578BDBM50438578(CHEMBL2413702)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438577BDBM50438577(CHEMBL2413703)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438570BDBM50438570(CHEMBL2413708)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438569BDBM50438569(CHEMBL2413709)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438572BDBM50438572(CHEMBL2413706)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438571BDBM50438571(CHEMBL2413707)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438570BDBM50438570(CHEMBL2413708)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438569BDBM50438569(CHEMBL2413709)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human tissue transglutaminase-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438579BDBM50438579(CHEMBL2413701)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438567BDBM50438567(CHEMBL512713)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438566BDBM50438566(CHEMBL2413711)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438574BDBM50438574(CHEMBL486969)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438572BDBM50438572(CHEMBL2413706)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438578BDBM50438578(CHEMBL2413702)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Aston University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50438577BDBM50438577(CHEMBL2413703)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human F13a-mediated biotin X-cadaverine incorporation into N,N'-dimethylcasein after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed