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Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50043279 Sort by
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)
Affinity DataIC50: 120nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)
Affinity DataIC50: 170nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)
Affinity DataIC50: 230nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Bovine)
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-amino-1,2-dihydroisoquinolin-1-one | CHEMBL44624...)
Affinity DataIC50: 250nMAssay Description:Inhibition of calf thymus PARP-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)
Affinity DataIC50: 260nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-amino-1,2-dihydroisoquinolin-1-one | CHEMBL44624...)
Affinity DataIC50: 300nMAssay Description:Inhibition of PARP-1 (unknown origin) in broken nuclear preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438608(CHEMBL2414049)
Affinity DataIC50: 320nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)
Affinity DataIC50: 330nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)
Affinity DataIC50: 480nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)
Affinity DataIC50: 490nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)
Affinity DataIC50: 570nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)
Affinity DataIC50: 730nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)
Affinity DataIC50: 830nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)
Affinity DataIC50: 880nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)
Affinity DataIC50: 900nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 2(Mouse)
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-amino-1,2-dihydroisoquinolin-1-one | CHEMBL44624...)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438606(CHEMBL2414052)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-amino-1,2-dihydroisoquinolin-1-one | CHEMBL44624...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438607(CHEMBL2414050)
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438609(CHEMBL2414047)
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed