Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50043329
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439441(CHEMBL2420738)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439440(CHEMBL2420739)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 1/2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50278299(1-(6-(7-chloroquinazolin-4-yloxy)pyridin-3-yl)-3-(...)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439442(CHEMBL2420737)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin) assessed as SUMO E1-SUMO thioester bond formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439436(CHEMBL2420740)
Affinity DataIC50: 3.54E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439439(CHEMBL1900956)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439437(CHEMBL1572155)
Affinity DataIC50: 3.57E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM50439438(CHEMBL1448459)
Affinity DataIC50: 5.73E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSUMO-activating enzyme subunit 2(Human)
Riken

Curated by ChEMBL
LigandPNGBDBM96736(MLS000860602 | SMR000458686 | cid_2814119 | N-{6-[...)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of SUMO E1 (unknown origin)-mediated RanGAP1 sumoylation by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed