Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50043389
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50310892(N,N'-(9-(2-(1-methylpyrrolidin-2-yl)ethylamino)acr...)
Affinity DataIC50: 18nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440391(CHEMBL2425367)
Affinity DataIC50: 28nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50134018(N-[9-(4-Amino-phenylamino)-6-(3-pyrrolidin-1-yl-pr...)
Affinity DataIC50: 60nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440390(ISOMETAMIDIUM)
Affinity DataIC50: 100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440389(CHEMBL1997011)
Affinity DataIC50: 100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440388(CHEMBL2425366)
Affinity DataIC50: 130nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440387(CHEMBL2425365)
Affinity DataIC50: 220nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50176906(N1-(10H-indolo[3,2-b]quinolin-11-yl)-N3,N3-dimethy...)
Affinity DataIC50: 440nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50111322(N,N-Dimethyl-N'-(11-nitro-13H-5,13-diaza-dibenzo[a...)
Affinity DataIC50: 500nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440386(CHEMBL2425364)
Affinity DataIC50: 750nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440385(CHEMBL2425363)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50068304(N-[9,10-Dioxo-6-(3-pyrrolidin-1-yl-propionylamino)...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440384(CHEMBL2425362)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50412201(Cryptolepine | CRYPTOLEPINE HYDROCHLORIDE)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440382(CHEMBL2425361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
Magna Graecia University of Catanzaro

Curated by ChEMBL
LigandPNGBDBM50440381(MERIDINE)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed