Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 6011
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104024(MK315)
Affinity DataIC50: 190nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104022(MK319)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM16238(IDD388 | {2-[(4-bromo-2-fluorobenzyl)carbamoyl]-5-...)
Affinity DataIC50: 400nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104020(MK181)
Affinity DataIC50: 710nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104021(MK408)
Affinity DataIC50: 1.19E+3nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104025(MK409)
Affinity DataIC50: 1.36E+3nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Human)
Academy of Sciences of The Czech Republic

LigandPNGBDBM104023(MK257)
Affinity DataIC50: 1.90E+3nMpH: 7.0 T: 2°CAssay Description:The assays were performed at 25 degrees Celsius in a 100mM sodium phosphate buffer (pH 7.0), with the AR protein amount reaching the Vmax and 0.2mM N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)