Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50043830
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446908(CHEMBL3115325)
Affinity DataIC50:  110nMAssay Description:Inhibition of JAK2 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446911(CHEMBL3112617)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446913(CHEMBL3115320)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446913(CHEMBL3115320)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of JAK2 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446908(CHEMBL3115325)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446911(CHEMBL3112617)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446910(CHEMBL3115323)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of JAK2 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446914(CHEMBL3115319)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446910(CHEMBL3115323)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446913(CHEMBL3115320)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446912(CHEMBL3115321)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446909(CHEMBL3115324)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446912(CHEMBL3115321)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446911(CHEMBL3112617)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446908(CHEMBL3115325)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of full-length ZAP70 (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446914(CHEMBL3115319)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50446909(CHEMBL3115324)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SYK (unknown origin) by radioactive ATP methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed