Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50005682
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192536BDBM192536(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192534BDBM192534(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192538BDBM192538(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50493599BDBM50493599(CHEMBL2436755)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192537BDBM192537(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192532BDBM192532(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192529BDBM192529(US9187480, ethyl N-{1-[8-(2-chlorophenyl)-9-(4-chl...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192535BDBM192535(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192531BDBM192531(US9187480, 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192533BDBM192533(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192536BDBM192536(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192535BDBM192535(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192537BDBM192537(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192529BDBM192529(US9187480, ethyl N-{1-[8-(2-chlorophenyl)-9-(4-chl...)
Affinity DataKi:  426nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192538BDBM192538(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  569nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192532BDBM192532(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  835nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192533BDBM192533(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192534BDBM192534(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.36E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 192531BDBM192531(US9187480, 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50493599BDBM50493599(CHEMBL2436755)
Affinity DataKi:  1.06E+4nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor (unknown origin) expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed