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Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50043794 Sort by
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50126186(2-(3-Naphthalen-2-yl-but-2-enoylamino)-benzoic aci...)
Affinity DataIC50: 93nMAssay Description:Inhibition of human telomerase isolated from human HeLa cells nuclear extracts expressed in insect cells assessed as [33P]dCMP incorporation after 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446424(U-73122 | CHEMBL1256678)
Affinity DataIC50: 200nMAssay Description:Inhibition of human telomerase activity in human Jurkat cells by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446426(CHEMBL3109742)
Affinity DataIC50: 400nMAssay Description:Inhibition of human telomerase activity after 8 mins by SYBR Green staining-based TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446421(CHEMBL3109740)
Affinity DataIC50: 470nMAssay Description:Inhibition of human telomerase isolated from human HeLa cells nuclear extracts expressed in insect cells assessed as [33P]dCMP incorporation after 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446422(Rel-Chrolactomycin | CHEMBL2164966)
Affinity DataIC50: 500nMAssay Description:Inhibition of human telomerase isolated from human A431 cellular extracts after 30 mins by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50396097(CHEMBL2170856)
Affinity DataIC50: 670nMAssay Description:Inhibition of human telomerase isolated from human U937 cellular extracts by SYBR Green staining-based TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446423(CHEMBL3109739)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human telomerase activity by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Rat)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50446425(CHEMBL3109741)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat telomerase by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50444911(CHEMBL3099733)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human telomerase isolated from human A431 cellular extracts after 30 mins by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50396098(CHEMBL2170857)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human telomerase activity by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed