Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50043444
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441236BDBM50441236(CHEMBL2431341)
Affinity DataKi:  2.10nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441235BDBM50441235(CHEMBL2431330)
Affinity DataKi:  2.80nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441237BDBM50441237(CHEMBL2431340)
Affinity DataKi:  3nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441241BDBM50441241(CHEMBL2431333 | CHEMBL2431336)
Affinity DataKi:  5nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441238BDBM50441238(CHEMBL2431339)
Affinity DataKi:  6.30nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441241BDBM50441241(CHEMBL2431333 | CHEMBL2431336)
Affinity DataKd:  7.80nMAssay Description:Binding affinity to PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441239BDBM50441239(CHEMBL2431338)
Affinity DataKi:  7.90nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441240BDBM50441240(CHEMBL2431337)
Affinity DataKi:  8.10nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265377BDBM50265377(CHEMBL496748 | CHEMBL2431335 | (S)-2-(3-((S)-1-Car...)
Affinity DataKd:  20nMAssay Description:Binding affinity to PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17659BDBM17659(pentanedioic acid analogue, (RS)-1 | 2-(phosphonom...)
Affinity DataKi:  31nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441234BDBM50441234(CHEMBL2431331)
Affinity DataKi:  62nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441233BDBM50441233(CHEMBL2431332)
Affinity DataKi:  95nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50441243BDBM50441243(CHEMBL2431334)
Affinity DataKd:  143nMAssay Description:Binding affinity to PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Kyoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102256BDBM50102256(2-[3-(1-Carboxy-2-mercapto-ethyl)-ureido]-pentaned...)
Affinity DataKi:  376nMAssay Description:Displacement of [123I]-DCIT from PSMA in human LNCaP cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed