Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50005748
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214615BDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataIC50: 0.794nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494136BDBM50494136(CHEMBL2441945)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494138BDBM50494138(CHEMBL2441946)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494137BDBM50494137(CHEMBL2441942)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494132BDBM50494132(CHEMBL2441941)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494141BDBM50494141(CHEMBL2441940)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494127BDBM50494127(CHEMBL2441944)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494135BDBM50494135(CHEMBL2441933)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494139BDBM50494139(CHEMBL2441938)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494131BDBM50494131(CHEMBL2441943)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494142BDBM50494142(CHEMBL2441935)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494130BDBM50494130(CHEMBL2441947)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494129BDBM50494129(CHEMBL2441948)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494128BDBM50494128(CHEMBL2441939)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494126BDBM50494126(CHEMBL2441949)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494134BDBM50494134(CHEMBL2441936)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494140BDBM50494140(CHEMBL2441934)
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494133BDBM50494133(CHEMBL2441937)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHO cells assessed as inhibition of forskolin/R-alpha-methylhistamine-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed