Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50043655
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084637BDBM50084637(Sivelestat | 2,2-Dimethyl-propionic acid 4-[2-(car...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444295BDBM50444295(CHEMBL3093806)
Affinity DataIC50: 80nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444297BDBM50444297(CHEMBL3093815)
Affinity DataIC50: 110nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444296BDBM50444296(CHEMBL3093814)
Affinity DataIC50: 180nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444300BDBM50444300(CHEMBL3093808)
Affinity DataIC50: 280nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444301BDBM50444301(CHEMBL3093809)
Affinity DataIC50: 300nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444312BDBM50444312(CHEMBL3093821)
Affinity DataIC50: 450nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444307BDBM50444307(CHEMBL3093816)
Affinity DataIC50: 670nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444302BDBM50444302(CHEMBL3093810)
Affinity DataIC50: 960nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444306BDBM50444306(CHEMBL3091487)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444305BDBM50444305(CHEMBL3093812)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084637BDBM50084637(Sivelestat | 2,2-Dimethyl-propionic acid 4-[2-(car...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human kallikrein using H-Pro-Phe-Arg-AMC acetate salt as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444299BDBM50444299(CHEMBL3093807)
Affinity DataIC50: 2.46E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444311BDBM50444311(CHEMBL3093820)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444304BDBM50444304(CHEMBL3093813)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444303BDBM50444303(CHEMBL3093811)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetMyeloblastin(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444297BDBM50444297(CHEMBL3093815)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444310BDBM50444310(CHEMBL3093819)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444309BDBM50444309(CHEMBL3093818)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444298BDBM50444298(CHEMBL3093805)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCathepsin G(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444295BDBM50444295(CHEMBL3093806)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate incubated for 30 mins prior to substrate addition measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetMyeloblastin(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444296BDBM50444296(CHEMBL3093814)
Affinity DataIC50: 4.75E+4nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444297BDBM50444297(CHEMBL3093815)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human kallikrein using H-Pro-Phe-Arg-AMC acetate salt as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444308BDBM50444308(CHEMBL3093817)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human neutrophil elastase using MeO-Suc-Ala-Ala-Pro-Val-AMC as substrate incubated for 30 mins prior to substrate addition measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444296BDBM50444296(CHEMBL3093814)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human kallikrein using H-Pro-Phe-Arg-AMC acetate salt as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444295BDBM50444295(CHEMBL3093806)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human kallikrein using H-Pro-Phe-Arg-AMC acetate salt as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCathepsin G(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444296BDBM50444296(CHEMBL3093814)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate incubated for 30 mins prior to substrate addition measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCathepsin G(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084637BDBM50084637(Sivelestat | 2,2-Dimethyl-propionic acid 4-[2-(car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate incubated for 30 mins prior to substrate addition measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetMyeloblastin(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444295BDBM50444295(CHEMBL3093806)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetMyeloblastin(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084637BDBM50084637(Sivelestat | 2,2-Dimethyl-propionic acid 4-[2-(car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCathepsin G(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50444297BDBM50444297(CHEMBL3093815)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate incubated for 30 mins prior to substrate addition measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed