Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50043663
TargetHexokinase-4(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444409(CHEMBL3091581)
Affinity DataIC50:  1.70E+3nMAssay Description:Activation of glucokinase in Wistar rat hepatocytes assessed as nuclear to cytosolic translocation of protein by immunofluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444410(CHEMBL3091580)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of glucokinase in rat INS-1 cells assessed as glucose-stimulated insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444411(CHEMBL3091585)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444412(CHEMBL3091584)
Affinity DataEC50:  1.35E+3nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444414(CHEMBL3091582)
Affinity DataEC50:  113nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444409(CHEMBL3091581)
Affinity DataEC50:  201nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444410(CHEMBL3091580)
Affinity DataEC50:  137nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444409(CHEMBL3091581)
Affinity DataEC50:  1.74E+5nMAssay Description:Activation of glucokinase in rat INS-1 cells assessed as glucose-stimulated insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50444413(CHEMBL3091583)
Affinity DataEC50:  227nMAssay Description:Activation of recombinant human glucokinase by G6PDH/NADP coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed