Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50043732
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataEC50:  8.13nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataIC50: 8.90nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445382(CHEMBL3104637)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445382(CHEMBL3104637)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445369(CHEMBL3104465)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445369(CHEMBL3104465)
Affinity DataEC50:  21nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445369(CHEMBL3104465)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445369(CHEMBL3104465)
Affinity DataEC50:  21nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataEC50:  22nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataEC50:  22nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445371(CHEMBL3104463)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445372(CHEMBL3104462)
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445371(CHEMBL3104463)
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445372(CHEMBL3104462)
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataEC50:  40nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataEC50:  41nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445381(CHEMBL3104638)
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445381(CHEMBL3104638)
Affinity DataIC50: 47nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445382(CHEMBL3104637)
Affinity DataEC50:  54nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445382(CHEMBL3104637)
Affinity DataEC50:  54nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445380(CHEMBL3104639)
Affinity DataIC50: 58nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445380(CHEMBL3104639)
Affinity DataIC50: 58nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445373(CHEMBL3104461)
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445373(CHEMBL3104461)
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445367(CHEMBL3104467)
Affinity DataIC50: 88nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445367(CHEMBL3104467)
Affinity DataIC50: 89nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445380(CHEMBL3104639)
Affinity DataEC50:  89nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445380(CHEMBL3104639)
Affinity DataEC50:  89.1nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445371(CHEMBL3104463)
Affinity DataEC50:  117nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445371(CHEMBL3104463)
Affinity DataEC50:  117nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445373(CHEMBL3104461)
Affinity DataEC50:  159nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445373(CHEMBL3104461)
Affinity DataEC50:  162nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445379(CHEMBL3104640)
Affinity DataIC50: 181nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445379(CHEMBL3104640)
Affinity DataIC50: 182nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445372(CHEMBL3104462)
Affinity DataEC50:  251nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Rat)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445372(CHEMBL3104462)
Affinity DataEC50:  251nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445377(CHEMBL3104643)
Affinity DataIC50: 277nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445377(CHEMBL3104643)
Affinity DataIC50: 282nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445375(CHEMBL3104459)
Affinity DataIC50: 361nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445375(CHEMBL3104459)
Affinity DataIC50: 363nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
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