Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50044283 Sort by
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50425555(CHEMBL2313653)
Affinity DataIC50: 400nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011368(CHEMBL3260989)
Affinity DataIC50: 600nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50326557(NSC45576, 2 | CHEMBL1253920 | (E)-5-((2-hydroxynap...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of EPAC1 (unknown origin) assessed as cAMP-mediated GEF activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011357(CHEMBL3260988)
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50: 7.00E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011358(CHEMBL1372282)
Affinity DataIC50: 7.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50384264(CHEMBL316966)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed