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Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50044283
TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50425555(CHEMBL2313653)
Affinity DataIC50:  400nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011368(CHEMBL3260989)
Affinity DataIC50:  600nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50326557((E)-5-((2-hydroxynaphthalen-1-yl)diazenyl)naphthal...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of EPAC1 (unknown origin) assessed as cAMP-mediated GEF activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011357(CHEMBL3260988)
Affinity DataIC50:  3.80E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataIC50:  7.00E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50011358(CHEMBL1372282)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of 8-NBD-cAMP from EPAC2 (unknown origin) by fluorescence plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRap guanine nucleotide exchange factor 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50384264(CHEMBL316966)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of EPAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)