Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50005795
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491950(CHEMBL2386692)
Affinity DataIC50:  821nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494500(CHEMBL3092720)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494501(CHEMBL3092721)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494503(CHEMBL3092723)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of thrombin (unknown origin) using z-Gly-Pro-Arg-4MbetaNA-acetate as substrate preincubated for 20 mins before substrate addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494502(CHEMBL3092722)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494503(CHEMBL3092723)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed