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Found 21 Enz. Inhib. hit(s) with all data for entry = 50043736
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445447(CHEMBL3104694)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at CCR5 (unknown origin) expressed in CHO cell membranes assessed as inhibition of RANTES-stimulated [35S]-GTPgammaS binding afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50334986(4,4-Difluoro-cyclohexanecarboxylic acid {(S)-3-[(1...)
Affinity DataIC50:  25nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445431(CHEMBL3104691)
Affinity DataIC50:  26nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445440(CHEMBL3104682)
Affinity DataIC50:  26nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445438(CHEMBL3104684)
Affinity DataIC50:  26nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445439(CHEMBL3104683)
Affinity DataIC50:  35nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445441(CHEMBL3104681)
Affinity DataIC50:  64nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445437(CHEMBL3104685)
Affinity DataIC50:  75nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445434(CHEMBL3104688)
Affinity DataIC50:  76nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445432(CHEMBL3104690)
Affinity DataIC50:  87nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445443(CHEMBL3104679)
Affinity DataIC50:  94nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445429(CHEMBL3104693)
Affinity DataIC50:  126nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445430(CHEMBL3104692)
Affinity DataIC50:  152nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445433(CHEMBL3104689)
Affinity DataIC50:  197nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445445(CHEMBL3104677)
Affinity DataIC50:  202nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445447(CHEMBL3104694)
Affinity DataIC50:  252nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445444(CHEMBL3104678)
Affinity DataIC50:  320nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445442(CHEMBL3104680)
Affinity DataIC50:  473nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445446(CHEMBL3104695)
Affinity DataIC50:  525nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445435(CHEMBL3104687)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50445436(CHEMBL3104686)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in CHO cells assessed as inhibition of RANTES-induced intracellular Ca2+ mobilization after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed