Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 6136
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111473BDBM111473(4-Methyl-N-(4-(2-morpholinoethoxy) phenyl)-3-(4-(p...)
Affinity DataIC50: 10nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111449BDBM111449(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 136nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111466BDBM111466(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 210nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 50237710BDBM50237710(AMN 107 | AMN107 | 4-methyl-N-[3-(4-methyl-1H-imid...)
Affinity DataIC50: 214nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111456BDBM111456(N-(3-bromo-5-(trifluoromethyl) phenyl)-4-methyl-3-...)
Affinity DataIC50: 219nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111455BDBM111455(N-(3,5-bis(trifluoromethyl) phenyl)-4-methyl-3-(4-...)
Affinity DataIC50: 259nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111465BDBM111465(N-(5-chloropyridin-2-yl)-4-methyl-3-(4-(pyridin-3-...)
Affinity DataIC50: 305nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111452BDBM111452(N-(4-bromophenyl)-4-methyl-3-(4-(pyridin-3-yl) pyr...)
Affinity DataIC50: 483nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111460BDBM111460(N-(3-acetylphenyl)-4-methyl-3-(4-(pyridin-3-yl) py...)
Affinity DataIC50: 542nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111453BDBM111453(N-(2-fluorophenyl)-4-methyl-3-(4-(pyridin-3-yl) py...)
Affinity DataIC50: 569nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111451BDBM111451(N-(4-methoxyphenyl)-4-methyl-3-(4-(pyridin-3-yl) p...)
Affinity DataIC50: 924nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111459BDBM111459(N-(2, 6-dimethylphenyl)-4-methyl-3-(4-(pyridin-3-y...)
Affinity DataIC50: 956nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111454BDBM111454(N-(3-fluorophenyl)-4-methyl-3-(4-(pyridin-3-yl) py...)
Affinity DataIC50: 1.07E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111457BDBM111457(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 1.11E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111450BDBM111450(N-(3, 4-dichlorophenyl)-4-methyl-3-(4-(pyridin-3-y...)
Affinity DataIC50: 1.51E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111462BDBM111462(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 2.19E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111464BDBM111464(4-Methyl-N-(pyridin-2-yl)-3-(4-(pyridin-3-yl) pyri...)
Affinity DataIC50: 3.58E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111467BDBM111467(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 3.58E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111463BDBM111463(4-Methyl-N-(pyridin-3-yl)-3-(4-(pyridin-3-yl) pyri...)
Affinity DataIC50: 4.03E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111461BDBM111461(N-(3-methoxyphenyl)-4-methyl-3-(4-(pyridin-3-yl) p...)
Affinity DataIC50: 5.24E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111448BDBM111448(N-(3-chloro-4-fluorophenyl)-4-methyl-3-(4-(pyridin...)
Affinity DataIC50: 9.57E+3nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111468BDBM111468(N-(4-(3-(dimethylamino)propoxy) phenyl)-4-methyl- ...)
Affinity DataIC50: 1.32E+4nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111469BDBM111469(N-(4-(2-(dimethylamino)ethoxy)phenyl)-4-methyl-3-(...)
Affinity DataIC50: 2.10E+4nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111474BDBM111474(4-Methyl-N-(4-(3-morpholinopropoxy) phenyl)-3-(4-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111472BDBM111472(4-Methyl-N-(4-(2-(piperidin-1-yl) ethoxy) phenyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111471BDBM111471(4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed
TargetBreakpoint cluster region protein [1-693](Human)
Xi'An Jiaotong University

LigandChemical structure of BindingDB Monomer ID 111470BDBM111470(N-(4-(2-(diethylamino)ethoxy)phenyl)-4-methyl-3-(4...)
Affinity DataIC50: 1.00E+5nMAssay Description:ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2014
Entry Details Article
PubMed