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Found 48 Enz. Inhib. hit(s) with all data for entry = 50043869
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447701(CHEMBL3113206)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447744(CHEMBL3112990)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447702(CHEMBL3112985)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50343449(CHEMBL1775171 | isopropyl 4-(1-(4-(methylsulfonyl)...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435635(CHEMBL2391601)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447703(CHEMBL3113003)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447704(CHEMBL3112989)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447705(CHEMBL3113016)
Affinity DataEC50:  860nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447706(CHEMBL3113014)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447707(CHEMBL3113009)
Affinity DataEC50:  590nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447708(CHEMBL3113006)
Affinity DataEC50:  550nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447709(CHEMBL3113008)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447710(CHEMBL3113007)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447711(CHEMBL3112996)
Affinity DataEC50:  310nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447712(CHEMBL3113004)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447713(CHEMBL3113207)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447714(CHEMBL3113005)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447715(CHEMBL3112983)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447716(CHEMBL3112980)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447717(CHEMBL3113010)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447718(CHEMBL3112986)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447719(CHEMBL3112979)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447720(CHEMBL3113205)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447721(CHEMBL3112981)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447722(CHEMBL3113011)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447723(CHEMBL3112997)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435643(CHEMBL2391593)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447724(CHEMBL3112995)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447725(CHEMBL3112988)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447726(CHEMBL3113019)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447727(CHEMBL3112999)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447728(CHEMBL3112998)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447729(CHEMBL3113017)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447730(CHEMBL3113013)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447731(CHEMBL3113012)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447732(CHEMBL3112993)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447733(CHEMBL3112991)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447734(CHEMBL3112987)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447735(CHEMBL3112982)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447736(CHEMBL3113015)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447737(CHEMBL3112992)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447738(CHEMBL3113018)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447739(CHEMBL3112994)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447740(CHEMBL3112984)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447741(CHEMBL3113000)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447742(CHEMBL3113002)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50447743(CHEMBL3113001)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50435665(CHEMBL2391602)
Affinity DataEC50:  310nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed