Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50043816
TargetTranscription factor Jun(Homo sapiens (Human))
National Defense Medical Center, Taiwan

Curated by ChEMBL
LigandPNGBDBM50446664(CHEMBL3113338)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of transcription factor AP-1 binding to oligonucleotide containing TPA-responsive element in TPA-activated human HeLa cells after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
National Defense Medical Center, Taiwan

Curated by ChEMBL
LigandPNGBDBM50446663(CHEMBL3113339)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of transcription factor AP-1 binding to oligonucleotide containing TPA-responsive element in TPA-activated human HeLa cells after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
National Defense Medical Center, Taiwan

Curated by ChEMBL
LigandPNGBDBM50446665(CHEMBL3112597)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of transcription factor AP-1 binding to oligonucleotide containing TPA-responsive element in TPA-activated human HeLa cells after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
National Defense Medical Center, Taiwan

Curated by ChEMBL
LigandPNGBDBM50133496((2R)-3-(3,4-dihydroxyphenyl)-2-[(2E)-3-(3,4-dihydr...)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of transcription factor AP-1 binding to oligonucleotide containing TPA-responsive element in TPA-activated human HeLa cells after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed