Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50044095
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001759(CHEMBL3233260)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001758(CHEMBL3233259)
Affinity DataIC50: 0.860nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001762(CHEMBL3233263)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 15nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001758(CHEMBL3233259)
Affinity DataIC50: 20nMAssay Description:Inhibition of LAP binding to human alphavbeta6 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001762(CHEMBL3233263)
Affinity DataIC50: 64nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001761(CHEMBL3233262)
Affinity DataIC50: 75nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001759(CHEMBL3233260)
Affinity DataIC50: 108nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001757(CHEMBL3233258)
Affinity DataIC50: 110nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001758(CHEMBL3233259)
Affinity DataIC50: 127nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001758(CHEMBL3233259)
Affinity DataIC50: 227nMAssay Description:Inhibition of vitronectin binding to alphavbeta5 integrin receptor (unknown origin) after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001760(CHEMBL3233261)
Affinity DataIC50: 638nMAssay Description:Inhibition of vitronectin binding to human alphavbeta3 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of fibrinogen binding to alpha2bbeta3 integrin receptor (unknown origin) after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001757(CHEMBL3233258)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001758(CHEMBL3233259)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of fibrinogen binding to alpha2bbeta3 integrin receptor (unknown origin) after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001759(CHEMBL3233260)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of fibrinogen binding to alpha2bbeta3 integrin receptor (unknown origin) after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001760(CHEMBL3233261)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Technische Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50001761(CHEMBL3233262)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of fibronectin binding to human alpha5beta1 integrin receptor after 1 hr by competitive solid-phase binding ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed