Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50044125
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004348(CHEMBL3237850)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004350(CHEMBL3237852)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004340(CHEMBL3237854)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004344(CHEMBL3237857)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004348(CHEMBL3237850)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004336(CHEMBL3237853)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004336(CHEMBL3237853)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004347(CHEMBL3237849)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004348(CHEMBL3237850)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004347(CHEMBL3237849)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004336(CHEMBL3237853)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004347(CHEMBL3237849)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004342(CHEMBL3237855)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004345(CHEMBL3237858)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004340(CHEMBL3237854)
Affinity DataIC50:  3.49E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004349(CHEMBL3237851)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004346(CHEMBL3237848)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004343(CHEMBL3237856)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004351(CHEMBL3233061)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004346(CHEMBL3237848)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004351(CHEMBL3233061)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004344(CHEMBL3237857)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004343(CHEMBL3237856)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004342(CHEMBL3237855)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004340(CHEMBL3237854)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004351(CHEMBL3233061)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004350(CHEMBL3237852)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004349(CHEMBL3237851)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004346(CHEMBL3237848)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004345(CHEMBL3237858)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004344(CHEMBL3237857)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004343(CHEMBL3237856)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004342(CHEMBL3237855)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004345(CHEMBL3237858)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004350(CHEMBL3237852)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM50004349(CHEMBL3237851)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Siedlce University Of Natural Sciences And Humanities

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed