Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50044326 Sort by
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013126(CHEMBL3261990)
Affinity DataKd:  2.26E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013133(CHEMBL3261987)
Affinity DataKd:  3.02E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013132(CHEMBL3261986)
Affinity DataKd:  5.23E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013130(CHEMBL3261985)
Affinity DataKd:  5.80E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013129(CHEMBL3261984)
Affinity DataKd:  4.29E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataKd:  2.19E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50011780(Pralidoxine chloride | PRALIDOXIME | CHEMBL748 | 2...)
Affinity DataKd:  3.14E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013120(CHEMBL3261992)
Affinity DataKd:  1.75E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013127(CHEMBL3261991)
Affinity DataKd:  5.49E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013125(CHEMBL3261989)
Affinity DataKd:  6.58E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013122(CHEMBL3261988)
Affinity DataKd:  1.69E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013133(CHEMBL3261987)
Affinity DataKd:  1.97E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013130(CHEMBL3261985)
Affinity DataKd:  8.89E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013129(CHEMBL3261984)
Affinity DataKd:  4.87E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataKd:  2.15E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013132(CHEMBL3261986)
Affinity DataKd:  8.61E+4nMAssay Description:Binding affinity to VX-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50011780(Pralidoxine chloride | PRALIDOXIME | CHEMBL748 | 2...)
Affinity DataKd:  2.57E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013120(CHEMBL3261992)
Affinity DataKd:  8.55E+3nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013127(CHEMBL3261991)
Affinity DataKd:  4.84E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013126(CHEMBL3261990)
Affinity DataKd:  2.08E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013122(CHEMBL3261988)
Affinity DataKd:  2.44E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013125(CHEMBL3261989)
Affinity DataKd:  8.43E+4nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataIC50: 8.70E+5nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013125(CHEMBL3261989)
Affinity DataIC50: 9.30E+5nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50011780(Pralidoxine chloride | PRALIDOXIME | CHEMBL748 | 2...)
Affinity DataIC50: 1.19E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013127(CHEMBL3261991)
Affinity DataIC50: 1.67E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013126(CHEMBL3261990)
Affinity DataIC50: 1.70E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013122(CHEMBL3261988)
Affinity DataIC50: 1.43E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013133(CHEMBL3261987)
Affinity DataIC50: 1.79E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013132(CHEMBL3261986)
Affinity DataIC50: 1.06E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013130(CHEMBL3261985)
Affinity DataIC50: 1.07E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013129(CHEMBL3261984)
Affinity DataIC50: 2.53E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Defence Research & Development Establishment (Drde)

Curated by ChEMBL
LigandPNGBDBM50013120(CHEMBL3261992)
Affinity DataIC50: 2.10E+6nMAssay Description:Inhibition of hemoglobin free human erythrocyte ghost acetylcholinesterase using acetylthiocholineiodide as substrate measured up to 1 hr by Ellman m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed