Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50044359
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014335(CHEMBL1164066)
Affinity DataIC50: 340nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014335(CHEMBL1164066)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014177(CHEMBL3221239)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014173(CHEMBL3260888)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014300(CHEMBL3260892)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014313(CHEMBL3260894)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014172(CHEMBL3221238)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014327(CHEMBL3221246)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014238(CHEMBL3260891)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014303(CHEMBL3260893)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014171(CHEMBL3221248)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014333(CHEMBL3221247)
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014300(CHEMBL3260892)
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014334(CHEMBL1164407)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014235(CHEMBL3221242)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014176(CHEMBL3221240)
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014178(CHEMBL3260889)
Affinity DataIC50: 2.84E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014179(CHEMBL3260890)
Affinity DataIC50: 2.98E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014317(CHEMBL3260895)
Affinity DataIC50: 4.41E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014328(CHEMBL3261115)
Affinity DataIC50: 5.55E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014257(CHEMBL3221244)
Affinity DataIC50: 5.62E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014321(CHEMBL3260896)
Affinity DataIC50: 5.71E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014248(CHEMBL3221243)
Affinity DataIC50: 5.96E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014333(CHEMBL3221247)
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014175(CHEMBL3221241)
Affinity DataIC50: 9.58E+4nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1D(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50014272(CHEMBL3221245)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human Cav1.3 channel in human SH-SY5Y cells assessed as 70 mM K+ induced calcium elevation compound treated 15 mins before stimulus by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed