Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50044374 Sort by
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50277889(CHEMBL451887 | CARFILZOMIB)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015247(CHEMBL3262766)
Affinity DataIC50: 110nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015246(CHEMBL3262765)
Affinity DataIC50: 170nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015242(CHEMBL3262758)
Affinity DataIC50: 190nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015240(CHEMBL3262756)
Affinity DataIC50: 220nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015236(CHEMBL3262752)
Affinity DataIC50: 340nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015239(CHEMBL3262755)
Affinity DataIC50: 340nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015241(CHEMBL3262757)
Affinity DataIC50: 360nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015238(CHEMBL3262754)
Affinity DataIC50: 380nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015237(CHEMBL3262753)
Affinity DataIC50: 440nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015244(CHEMBL3262762)
Affinity DataIC50: 630nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-7(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50015243(CHEMBL3262761)
Affinity DataIC50: 950nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed