Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50044476
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007207BDBM50007207(CHEMBL3237860)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007208BDBM50007208(CHEMBL3237861)
Affinity DataIC50: 29nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430990BDBM50430990(BELACTOSIN A)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018677BDBM50018677(CHEMBL3291290)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018678BDBM50018678(CHEMBL3291291)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed