Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50044503 Sort by
TargetP2Y purinoceptor 1(Human)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  850nMAssay Description:Agonist activity at human P2Y1 receptor expressed in human 1321N1 cells assessed as increase of intracellular calcium level after 30 mins using fura-...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 11(Human)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50019292(CHEMBL3289393)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human P2Y11 receptor expressed in human 1321N1 cells assessed as increase of intracellular calcium level after 30 mins using fura...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019296(CHEMBL3289396)
Affinity DataIC50: 390nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019294(CHEMBL3289394)
Affinity DataIC50: 600nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019291(CHEMBL3289392)
Affinity DataIC50: 1.63E+4nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019292(CHEMBL3289393)
Affinity DataIC50: 1.87E+4nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019295(CHEMBL3289395)
Affinity DataIC50: 3.12E+4nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019296(CHEMBL3289396)
Affinity DataKi:  20nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019294(CHEMBL3289394)
Affinity DataKi:  685nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019292(CHEMBL3289393)
Affinity DataKi:  1.30E+3nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019291(CHEMBL3289392)
Affinity DataKi:  4.50E+3nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019291(CHEMBL3289392)
Affinity DataKi:  4.50E+3nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate assessed as dissociation constant for enzyme-inhibitor-substrate complex after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019295(CHEMBL3289395)
Affinity DataKi:  1.52E+4nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate after 20 mins by Dixon and Cornish-Bowden methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50019295(CHEMBL3289395)
Affinity DataKi:  1.92E+5nMAssay Description:Mixed type inhibition of human NPP1 using pNP-TMP as substrate assessed as dissociation constant for enzyme-inhibitor-substrate complex after 20 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed