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Found 10 Enz. Inhib. hit(s) with all data for entry = 50044414
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016496(CHEMBL3260241)
Affinity DataIC50:  30nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016508(CHEMBL3260249)
Affinity DataIC50:  90nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016502(CHEMBL3260248)
Affinity DataIC50:  120nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016495(CHEMBL3260236)
Affinity DataIC50:  190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016501(CHEMBL3260247)
Affinity DataIC50:  190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016498(CHEMBL3260243)
Affinity DataIC50:  590nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016500(CHEMBL3260246)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016497(CHEMBL3260242)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016499(CHEMBL3260244)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016509(CHEMBL3260250)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed