Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50043773
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Inhibition of recombinant LSD1 (178 to 831) (unknown origin) expressed in baculovirus infected insect Sf9 cells using diMeK4H3-21 as substrate by per...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of human recombinant LSD1 using di-methylated H3-K4 peptide as substrate assessed as release of H2O2 preincubated for 15 mins followed by ...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of human recombinant LSD1 using di-methylated H3-K4 peptide as substrate assessed as release of H2O2 preincubated for 15 mins followed by ...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using methylated H3-K4 peptide as substrate by peroxidase-coupled assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1 [4-485](Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of recombinant human LSD1/CoREST complex expressed in Escherichia coli using methylated H3-K4 peptide as substrate by peroxidase-coupled a...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Inhibition of recombinant LSD1 (178 to 831) (unknown origin) expressed in baculovirus infected insect Sf9 cells using diMeK4H3-21 as substrate by per...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of recombinant LSD1 (unknown origin) using di-methylated H3-K4 peptide as substrate incubated for 5 mins prior to substrate addition by fl...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 385nMAssay Description:Competitive inhibition of recombinant LSD1 (unknown origin) using H3K4Me2 peptide as substrate preincubated for 30 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Competitive inhibition of recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using H3K4 peptide as substrate by Dixon p...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant LSD1 (unknown origin) using di-methylated H3-K4 peptide as substrate incubated for 5 mins prior to substrate addition by fl...More data for this Ligand-Target Pair
