Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50040352
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 160nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 300nMAssay Description:Inhibition of EphB4 by FRET assay in presence of 30 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 338nMAssay Description:Inhibition of recombinant Src catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 864nMAssay Description:Inhibition of recombinant Abl1 catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 930nMAssay Description:Inhibition of human full length EphB4 expressed in MEF cells assessed as inhibition of human ephrin B2/FC chimera-stimulated receptor autophosphoryla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of recombinant Lck catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393034BDBM50393034(CHEMBL2152704)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of recombinant EGFR catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393033BDBM50393033(CHEMBL2152699)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393035BDBM50393035(CHEMBL2152698)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393033BDBM50393033(CHEMBL2152699)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of EphB4 by FRET assay in presence of 30 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393036BDBM50393036(CHEMBL2152702)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed