Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50040464
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394591BDBM50394591(CHEMBL2164207)
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394596BDBM50394596(CHEMBL2164202)
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394588BDBM50394588(CHEMBL2164210)
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394601BDBM50394601(CHEMBL2164217)
Affinity DataIC50: 0.110nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394593BDBM50394593(CHEMBL2164205)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394592BDBM50394592(CHEMBL2164206)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394595BDBM50394595(CHEMBL2164203)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394587BDBM50394587(CHEMBL2164211)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394599BDBM50394599(CHEMBL2164219)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394598BDBM50394598(CHEMBL2164220)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394589BDBM50394589(CHEMBL2164209)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394590BDBM50394590(CHEMBL2164208)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394586BDBM50394586(CHEMBL2164212)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394603BDBM50394603(CHEMBL2164215)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394597BDBM50394597(CHEMBL2164201)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394600BDBM50394600(CHEMBL2164218)
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394605BDBM50394605(CHEMBL2164213)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359492BDBM50359492(CHEMBL1926888)
Affinity DataIC50: 10.9nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394602BDBM50394602(CHEMBL2164216)
Affinity DataIC50: 14.3nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394604BDBM50394604(CHEMBL2164214)
Affinity DataIC50: 31.1nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394594BDBM50394594(CHEMBL2164204)
Affinity DataIC50: 48.4nMAssay Description:Antagonist activity at CCR5 receptor expressed in P4R5 cells co-expressing CD4, and LTR-beta-gal construct assessed as inhibition of infusion to HIV ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394591BDBM50394591(CHEMBL2164207)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394595BDBM50394595(CHEMBL2164203)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394592BDBM50394592(CHEMBL2164206)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394599BDBM50394599(CHEMBL2164219)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394588BDBM50394588(CHEMBL2164210)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394598BDBM50394598(CHEMBL2164220)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394590BDBM50394590(CHEMBL2164208)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394587BDBM50394587(CHEMBL2164211)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50394586BDBM50394586(CHEMBL2164212)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant hERG expressed in CHO cells by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed