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Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50040066
TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388788(CHEMBL2062566)
Affinity DataIC50:  4nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388805(CHEMBL2062571)
Affinity DataIC50:  4nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388794(CHEMBL2062579)
Affinity DataIC50:  7nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388786(CHEMBL2062563)
Affinity DataIC50:  10nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388785(CHEMBL2062577)
Affinity DataIC50:  11nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388787(CHEMBL2062570)
Affinity DataIC50:  16nMAssay Description:Inhibition of CK2alpha in human DLD-1 cells assessed as decrease in AKT phosphorylation at S129 residue after 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388792(CHEMBL2062576)
Affinity DataIC50:  18nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50388783(CHEMBL2062565)
Affinity DataIC50:  20nMAssay Description:Inhibition of HipK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388787(CHEMBL2062570)
Affinity DataIC50:  24nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388782(CHEMBL2062564)
Affinity DataIC50:  26nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388778(CHEMBL2062580)
Affinity DataIC50:  27nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50388786(CHEMBL2062563)
Affinity DataIC50:  30nMAssay Description:Inhibition of HipK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388790(CHEMBL2062573)
Affinity DataIC50:  30nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388806(CHEMBL2062572)
Affinity DataIC50:  30nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388784(CHEMBL2062575)
Affinity DataIC50:  30nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388785(CHEMBL2062577)
Affinity DataIC50:  34nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388791(CHEMBL2062574)
Affinity DataIC50:  40nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50388782(CHEMBL2062564)
Affinity DataIC50:  50nMAssay Description:Inhibition of HipK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388800(CHEMBL2062561)
Affinity DataIC50:  52nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388805(CHEMBL2062571)
Affinity DataIC50:  57nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388797(CHEMBL2062557)
Affinity DataIC50:  58nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50388784(CHEMBL2062575)
Affinity DataIC50:  60nMAssay Description:Inhibition of HipK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388776(CHEMBL2062581)
Affinity DataIC50:  77nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388799(CHEMBL2062560)
Affinity DataIC50:  78nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388804(CHEMBL2062569)
Affinity DataIC50:  79nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388794(CHEMBL2062579)
Affinity DataIC50:  83nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCytochrome P450 1A2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388786(CHEMBL2062563)
Affinity DataIC50:  100nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388795(CHEMBL2062555)
Affinity DataIC50:  100nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388793(CHEMBL2062578)
Affinity DataIC50:  120nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388786(CHEMBL2062563)
Affinity DataIC50:  130nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388796(CHEMBL2062556)
Affinity DataIC50:  180nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388806(CHEMBL2062572)
Affinity DataIC50:  190nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388780(CHEMBL2062583)
Affinity DataIC50:  210nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388803(CHEMBL2062568)
Affinity DataIC50:  240nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388776(CHEMBL2062581)
Affinity DataIC50:  250nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388801(CHEMBL2062562)
Affinity DataIC50:  250nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388802(CHEMBL2062567)
Affinity DataIC50:  270nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388798(CHEMBL2062558)
Affinity DataIC50:  430nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388789(CHEMBL2062559)
Affinity DataIC50:  460nMAssay Description:Inhibition of full length N-terminus His-tagged human CK2alpha expressed in insect Sf21 cells using BODIPY-FL-RRRDDDSDDD-CONH2 as substrate after 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388790(CHEMBL2062573)
Affinity DataIC50:  460nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388779(CHEMBL2062582)
Affinity DataIC50:  500nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50388781(CHEMBL2062585)
Affinity DataIC50:  570nMAssay Description:Inhibition of HipK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388782(CHEMBL2062564)
Affinity DataIC50:  700nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388791(CHEMBL2062574)
Affinity DataIC50:  780nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388793(CHEMBL2062578)
Affinity DataIC50:  830nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388792(CHEMBL2062576)
Affinity DataIC50:  860nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388783(CHEMBL2062565)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCasein kinase II subunit alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388784(CHEMBL2062575)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of CK2alpha in human HCT116 cells assessed as decrease in AKT phosphorylation at S129 residue after 3 to 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388785(CHEMBL2062577)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlycogen synthase kinase-3 beta(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50388784(CHEMBL2062575)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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