Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50043612
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  900nMAssay Description:Agonist activity at GPR39 in human HT-29 cells assessed as increase in intracellular Ca2+ mobilization after 72 hrs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443617(CHEMBL3092410)
Affinity DataEC50:  840nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443618(CHEMBL3092411)
Affinity DataEC50:  310nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443619(CHEMBL3092412)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  56nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443617(CHEMBL3092410)
Affinity DataEC50:  190nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443618(CHEMBL3092411)
Affinity DataEC50:  320nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443619(CHEMBL3092412)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 39(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed