BindingDB PrimarySearch

Found 6 Enz. Inhib. hit(s) with all data for entry = 50043675

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM21675((4R)-4-[(1S,2S,5R,7S,8R,9R,10S,11S,14R,15R)-8-ethy...)

EC50: 100nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM50444530(CHEMBL3098607)

EC50: 1.32E+3nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM50236238((3alpha,5beta)-3-hydroxycholan-24-oic acid | 3alph...)

EC50: 730nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM21680((4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R,16S)-5,9,1...)

EC50: 1.98E+4nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM50300199(6alpha-ethyl-23(S)-methyl-cholic acid | CHEMBL5676...)

EC50: 180nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair

G-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

BDBM21674((4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R)-5,9-dihyd...)

EC50: 1.03E+4nMAssay Description:Agonist activity at wild type TGR5 (unknown origin)More data for this Ligand-Target Pair