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Found 14 Enz. Inhib. hit(s) with all data for entry = 50043608
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human c-Met using KKKSPGEYVNIEFG peptide as substrate by nanoliter kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443563(CHEMBL3091721)
Affinity DataIC50:  12nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443565(CHEMBL3091724)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  22nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443564(CHEMBL3091722)
Affinity DataIC50:  23nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  29nMAssay Description:Inhibition of human AXL (unknown origin) using EAIYAAPFAKKK peptide as substrate by nanoliter kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  39nMAssay Description:Inhibition of NPM-fused ALK phosphorylation (unknown origin) expressed in human karpas 299 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50:  110nMAssay Description:Inhibition of NPM-fused ALK phosphorylation (unknown origin) expressed in human karpas 299 cells after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443561(CHEMBL3091719)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443562(CHEMBL3091720)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Met phosphorylation in human MKN845 cells after 1 hr by western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50443560(CHEMBL3091723)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of full-length AXL (unknown origin) phosphorylation expressed in MEF after 90 mins by Sandwich-ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed