Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50043777
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446191(CHEMBL3109036)
Affinity DataIC50:  5nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446197(CHEMBL3109042)
Affinity DataIC50:  6nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446195(CHEMBL3109040)
Affinity DataIC50:  7nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446196(CHEMBL3109041)
Affinity DataIC50:  7nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446204(CHEMBL3109055)
Affinity DataIC50:  11nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446207(CHEMBL3109051)
Affinity DataIC50:  17nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446205(CHEMBL3109049)
Affinity DataIC50:  18nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446201(CHEMBL3109046)
Affinity DataIC50:  25nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446199(CHEMBL3109044)
Affinity DataIC50:  33nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446198(CHEMBL3109043)
Affinity DataIC50:  40nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446200(CHEMBL3109045)
Affinity DataIC50:  45nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446203(CHEMBL3109048)
Affinity DataIC50:  46nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446208(CHEMBL3109052)
Affinity DataIC50:  47nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446202(CHEMBL3109047)
Affinity DataIC50:  52nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446210(CHEMBL3109054)
Affinity DataIC50:  52nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446206(CHEMBL3109050)
Affinity DataIC50:  52nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446193(CHEMBL3109038)
Affinity DataIC50:  57nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446209(CHEMBL3109053)
Affinity DataIC50:  140nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446192(CHEMBL3109037)
Affinity DataIC50:  177nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Pharma Research

Curated by ChEMBL
LigandPNGBDBM50446194(CHEMBL3109039)
Affinity DataIC50:  5.76E+3nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with biotinylated p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed