Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50044275
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011209(CHEMBL3260324)
Affinity DataIC50: 5nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011201(CHEMBL3260326)
Affinity DataIC50: 6nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011202(CHEMBL3260325)
Affinity DataIC50: 9nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011188(CHEMBL3260329)
Affinity DataIC50: 30nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011200(CHEMBL3260327)
Affinity DataIC50: 500nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011189(CHEMBL3260328)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed