Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50044258 Sort by
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50004952(CHEMBL31344 | 3-(2-Carboxy-ethyl)-4,6-dichloro-1H-...)
Affinity DataKd:  1.26E+3nMAssay Description:Binding affinity to human GPR17 expressed in CHO-K1 cell membranes after 60 mins by saturation curve studyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50004952(CHEMBL31344 | 3-(2-Carboxy-ethyl)-4,6-dichloro-1H-...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by homologous competition binding assay in presence o...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50010475(GV-150526X | GAVESTINEL)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by heterologous competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50004952(CHEMBL31344 | 3-(2-Carboxy-ethyl)-4,6-dichloro-1H-...)
Affinity DataKi:  2.32E+3nMAssay Description:Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50023198(CHEMBL21333 | N-(4-oxo-2-(1H-tetrazol-5-yl)-4H-chr...)
Affinity DataKi:  4.06E+3nMAssay Description:Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by heterologous competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50052024(montelukast | CHEMBL787)
Affinity DataKi:  6.54E+3nMAssay Description:Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO-K1 cell membranes after 60 mins by heterologous competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed