TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human ACE C-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of human ACE N-terminal domain using Cbz-Phe-His-Leu-OH substrateMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of ACE (unknown origin)More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of rabbit lung somatic ACE using FAPGG substrateMore data for this Ligand-Target Pair
TargetDipeptidyl carboxypeptidase(Escherichia coli (strain K12))
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Vanderbilt University Department Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of Escherichia coli dipeptidyl carboxypeptidase assessed as FAPGG substrate hydrolysisMore data for this Ligand-Target Pair