Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50044263
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029(CHEMBL13470 | 3-[(4-Allyl-2,5-dimethyl-piperazin-1...)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  0.313nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  0.390nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  0.534nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  0.980nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029(CHEMBL13470 | 3-[(4-Allyl-2,5-dimethyl-piperazin-1...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human kappa opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029(CHEMBL13470 | 3-[(4-Allyl-2,5-dimethyl-piperazin-1...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029(CHEMBL13470 | 3-[(4-Allyl-2,5-dimethyl-piperazin-1...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human kappa opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010659(CHEMBL3264748)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010654(CHEMBL3264744)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010658(CHEMBL3264747)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010654(CHEMBL3264744)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human kappa opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010657(CHEMBL3264746)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010651(CHEMBL3264741)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010656(CHEMBL3264745)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010652(CHEMBL3264742)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50010653(CHEMBL3264743)
Affinity DataEC50:  113nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
Displayed 1 to 50 (of 71 total ) | Next | Last >>
Jump to: