Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50044271
TargetSodium- and chloride-dependent glycine transporter 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataEC50:  5nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataEC50:  10nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011136BDBM50011136(CHEMBL3259926)
Affinity DataEC50:  24nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011137BDBM50011137(CHEMBL3259935)
Affinity DataEC50:  25nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011138BDBM50011138(CHEMBL3259930)
Affinity DataEC50:  26nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011139BDBM50011139(CHEMBL3259931)
Affinity DataEC50:  28nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011140BDBM50011140(CHEMBL3259934)
Affinity DataEC50:  48nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011141BDBM50011141(CHEMBL3259937)
Affinity DataEC50:  54nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011142BDBM50011142(CHEMBL3259938)
Affinity DataEC50:  60nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011143BDBM50011143(CHEMBL3259925)
Affinity DataEC50:  67nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011144BDBM50011144(CHEMBL3259936)
Affinity DataEC50:  110nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011166BDBM50011166(CHEMBL3259943)
Affinity DataIC50: 140nMAssay Description:Inhibition of GlyT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011145BDBM50011145(CHEMBL3259933)
Affinity DataEC50:  170nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011146BDBM50011146(CHEMBL3259927)
Affinity DataEC50:  180nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011147BDBM50011147(CHEMBL3259939)
Affinity DataEC50:  180nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011149BDBM50011149(CHEMBL3259909)
Affinity DataEC50:  230nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011150BDBM50011150(CHEMBL3259910)
Affinity DataEC50:  230nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011151BDBM50011151(CHEMBL3259932)
Affinity DataEC50:  230nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011152BDBM50011152(CHEMBL3259911)
Affinity DataEC50:  270nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011153BDBM50011153(CHEMBL3259924)
Affinity DataEC50:  300nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011154BDBM50011154(CHEMBL3259923)
Affinity DataEC50:  320nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011155BDBM50011155(CHEMBL3259912)
Affinity DataEC50:  380nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011156BDBM50011156(CHEMBL3259919)
Affinity DataEC50:  540nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011157BDBM50011157(CHEMBL3259908)
Affinity DataEC50:  660nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011158BDBM50011158(CHEMBL3259929)
Affinity DataEC50:  670nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011159BDBM50011159(CHEMBL3259917)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011160BDBM50011160(CHEMBL3259940)
Affinity DataEC50:  1.67E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011161BDBM50011161(CHEMBL3259942)
Affinity DataEC50:  1.70E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011162BDBM50011162(CHEMBL3259918)
Affinity DataEC50:  4.80E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011164BDBM50011164(CHEMBL3259913)
Affinity DataEC50:  6.70E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011165BDBM50011165(CHEMBL3259922)
Affinity DataEC50:  9.90E+3nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011167BDBM50011167(CHEMBL3259914)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011173BDBM50011173(CHEMBL3259941)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011168BDBM50011168(CHEMBL3259915)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011169BDBM50011169(CHEMBL3259916)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011171BDBM50011171(CHEMBL3259920)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011172BDBM50011172(CHEMBL3259921)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human GlyT1 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of human GlyT2 expressed in cells assessed as [3H]glycine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50011135BDBM50011135(CHEMBL3259928)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed