Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50039692 Sort by
LigandPNGBDBM50382408(CHEMBL2022554)
Affinity DataIC50: 6.10E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50382406(CHEMBL1606364)
Affinity DataIC50: 9.80E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382405(CHEMBL2022172)
Affinity DataIC50: 1.44E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382406(CHEMBL1606364)
Affinity DataIC50: 1.96E+4nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382407(CHEMBL1536503)
Affinity DataIC50: 2.06E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382405(CHEMBL2022172)
Affinity DataIC50: 4.63E+4nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382408(CHEMBL2022554)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50382407(CHEMBL1536503)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed