Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50044563
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020865BDBM50020865(CHEMBL3286988)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020859BDBM50020859(CHEMBL3286982)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020860BDBM50020860(CHEMBL3286983)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020861BDBM50020861(CHEMBL3286984)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020867BDBM50020867(CHEMBL3286989)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020862BDBM50020862(CHEMBL3286985)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020858BDBM50020858(CHEMBL3286981)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020865BDBM50020865(CHEMBL3286988)
Affinity DataIC50: 6nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020859BDBM50020859(CHEMBL3286982)
Affinity DataIC50: 7nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020864BDBM50020864(CHEMBL3286987)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020869BDBM50020869(CHEMBL3286990)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020861BDBM50020861(CHEMBL3286984)
Affinity DataIC50: 18nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020862BDBM50020862(CHEMBL3286985)
Affinity DataIC50: 18nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020864BDBM50020864(CHEMBL3286987)
Affinity DataIC50: 32nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020860BDBM50020860(CHEMBL3286983)
Affinity DataIC50: 32nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020863BDBM50020863(CHEMBL3286986)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant human microtubule associated protein tau aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020858BDBM50020858(CHEMBL3286981)
Affinity DataIC50: 93nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020867BDBM50020867(CHEMBL3286989)
Affinity DataIC50: 123nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020869BDBM50020869(CHEMBL3286990)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Temple University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020863BDBM50020863(CHEMBL3286986)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of amyloid beta (unknown origin) aggregation by Thiazin-red R displacement fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed