Found 13 Enz. Inhib. hit(s) with all data for entry = 50045134 TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 60 mM K+-induced contractionMore data for this Ligand-Target Pair
3D Structure (crystal)TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 481nMAssay Description:Inhibition of L-type calcium channel in Wistar rat aorta rings assessed as reduction in L-type Ba(2+) current at Vh of -50 mVMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of L-type calcium channel in endothelium-intact Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 60 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-intact Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-intact Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 7.94E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 60 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rattus norvegicus)
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Vietnam Academy Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 2.51E+5nMAssay Description:Inhibition of L-type calcium channel in Wistar rat aorta rings assessed as reduction in L-type Ba(2+) current at Vh of -50 mVMore data for this Ligand-Target Pair
