Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50045177
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048413BDBM50048413(CHEMBL2370064)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001447BDBM50001447(His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu-Met-NH2(Neurok...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048411BDBM50048411(CHEMBL3360196)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048410BDBM50048410(CHEMBL3360197)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048409BDBM50048409(CHEMBL3360198)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048408BDBM50048408(CHEMBL3360199)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048415BDBM50048415(CHEMBL3360194)
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]SDF1 from CXCR4 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048406BDBM50048406(CHEMBL3360201)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048414BDBM50048414(CHEMBL3360195)
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125I]SDF1 from CXCR4 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048407BDBM50048407(CHEMBL3360200)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048405BDBM50048405(CHEMBL3360202)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed