Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50044590
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7533BDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021612BDBM50021612(CHEMBL3291228)
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021604BDBM50021604(CHEMBL3290949)
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021607BDBM50021607(CHEMBL3291224)
Affinity DataIC50: 730nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021611BDBM50021611(CHEMBL3291227)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021605BDBM50021605(CHEMBL3290950)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021609BDBM50021609(CHEMBL3291226)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021596BDBM50021596(CHEMBL3291232)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021597BDBM50021597(CHEMBL3291233)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021598BDBM50021598(CHEMBL3291234)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021599BDBM50021599(CHEMBL3286445)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021594BDBM50021594(CHEMBL3291230)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021595BDBM50021595(CHEMBL3291231)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021600BDBM50021600(CHEMBL3291235)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021608BDBM50021608(CHEMBL3291225)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021603BDBM50021603(CHEMBL3291236)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021606BDBM50021606(CHEMBL3291223)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed