Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50045315
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056344(CHEMBL3322514)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056343(CHEMBL3322513)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056349(CHEMBL3322507)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056350(CHEMBL3322508)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056347(CHEMBL3322502)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 4(Mouse)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at mouse LPA4 expressed in CHO cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human LPA1 expressed in LPA1xLPA2 double knockout mouse MEF cells up to 10 uM by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  510nMAssay Description:Agonist activity at FLAG-tagged human LPA5 expressed in rat B103 cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at human LPA3 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056348(CHEMBL3322503)
Affinity DataEC50:  1.42E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056346(CHEMBL3322501)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056345(CHEMBL3322500)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056342(CHEMBL3322509)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50056345(CHEMBL3322500)
Affinity DataIC50: 6.60E+3nMAssay Description:Antagonist activity at human LPA3 expressed in LPA1xLPA2 double knockout mouse MEF cells assessed as reduction in LP18:1-induced calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed